• A 419259 trihydrochloride
  • 3914-10mg
  • 10mg
Inhibitor of Src family kinases (SFK) (IC50 = 0.1 - 0.3 μM). Suppresses proliferation and induces apoptosis in CML cell lines including CD34+. Blocks Stat5 and Erk activation in vivo. Displays no inhibition of EGFR kinase activity in HNSCC cells.

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